Cart
sales@molnova.com
PKC-theta inhibitor(b)
CAS No. ——
PKC-theta inhibitor(b)( —— )
Catalog No. M20506 CAS No. ——
PKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 134 | Get Quote |
|
| 5MG | 268 | Get Quote |
|
| 10MG | 431 | Get Quote |
|
| 25MG | 853 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NamePKC-theta inhibitor(b)
-
NoteResearch use only, not for human use.
-
Brief DescriptionPKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM).
-
DescriptionPKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM).
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayAngiogenesis
-
TargetPKC
-
RecptorPKCθ
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number——
-
Formula Weight454.4
-
Molecular FormulaC20H25F3N6O3?
-
Purity>98% (HPLC)
-
SolubilityDMSO:62.5 mg/mL?(137.53 mM)
-
SMILESCl.NCC1CCC(CNc2nc(NCc3ccccc3OC(F)(F)F)ncc2[N+]([O-])=O)CC1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Cywin C L Dahmann G Iii A S P et al. Discovery of potent and selective PKC-θ inhibitors[J]. Bioorganic & Medicinal Chemistry Letters 2007 17(1):225-230.
molnova catalog
related products
-
PKCiota-IN-49
PKCiota-IN-49 is a potent and selective inhibitor of Protein Kinase C iota (PKC-ι) with IC50 of 2.8 nM.
-
Pep2m, myristoylated
Cell-permeable, myristoylated form of pep2m. Peptide inhibitor of the interaction between the C-terminus of the GluA2 (AMPA receptor) subunit and N-ethylmaleimide-sensitive fusion protein (NSF), a protein that regulates AMPA receptor function. Reduces postsynaptic currents in CA1 neurons, AMPA-mediated currents in cultured hippocampal neurons and AMPA receptor surface expression.
-
Solamargine
Solamargine is a major steroidal alkaloid glycoside extracted from a traditional Chinese medicine herb, Solanum nigrum L. (SNL); has been shown to inhibit growth and induce apoptosis of various cancer cells.
